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康贵峰

姓名:康贵峰

性别:男

职称:讲师

 

招生院所:药学院

招生类型:

招生专业:药物化学

研究方向名称:药物化学,有机化学

电子信箱:guifengkang@qq.com

个人简介

2016年进入多肽及小分子药物北京市重点实验室,任药物化学系讲师。讲授课程包括药物化学、有机化学、药物的波谱解析实验、专业药学实验等。

研究方向为杂环小分子的设计、合成、活性评价及作用机制研究。

 

教育经历

2005/8 - 2008/7,北京大学药学院,博士,导师:彭师奇、赵明。

2002/9 - 2005/7,中国科学院山西煤化所,硕士,导师:王建国。

1998/9 - 2002/7,西北大学化学系,学士。

 

工作经历

2016/1 - 至今,首都医科大学化学生物学院药学院,教师

2014/9 - 2015/12,美国弗吉尼亚联邦大学药物化学系,博士后

2012/4 - 2013/11,北京四环制药,项目经理

2009/12 - 2014/1,浙江大学、浙江医药股份有限公司新昌制药厂联合培养,博士后

2009/12 - 2012/3,浙江医药股份有限公司新昌制药厂,职工

2008/9 - 2009/10,康龙化成(北京)新药技术有限公司,高级研究员

 

重要学术论文

1. Guifeng Kang, Yuji Wang, Jiawang Liu, Jianhui Wu, Ming Zhao, Guochun Li, Ning Li, Li Peng, Xiaoyi Zhang, Li Li, Nathan Mair, Shiqi Peng, Development of three-component conjugates : to get nano-globes with pouous surfaces, high in vivo anti-osteoporosis activity and minimal side effects, J.Mater. Chem.,09/ 2012, 22(40), 21740-21748.

2. Guifeng Kang, Ming Zhao, Xiaoyi Zhang, Li Peng, Chunbo Li, Wei Mao, Weidong Ye, Shiqi Peng “A class of novel conjugates of substituted purine and Gly-AA-OBzl: Synthesis and evaluation of orally analgesic activity”, Bioorg. Med. Chem. Lett.,10/2010, 20(20), 6157-6160.

3. Yuji Wang, Guifeng Kang, Jiawang Liu, Ming Zhao, Jianhui Wu, Xiaoyi Zhang, Ye Li, Xiaobo Zhong, Yifan Yang, Shiqi Peng, Novel potassium N-[(2S, 3R, 4R, 5R)-2,3,4,5,6-pentahy -droxylhex-1-yl]-L-amino acid dichloroplatinates(II) with high anti-tumor activity and low side reaction, Metallomics, 04/2012, 4(5), 441-447.

4. Jinghua Zhao, Guifeng Kang, Wei Wang, Ming Zhao, Xiaoyi Zhang, Chunbo Lu, Wei Mao, Heng Wei Chang, Weidong Ye, Shiqi Peng, N-[2-Chloro-9H-purin-6-yl]-N- cyclopropylgly- cylamino acids and derivatives: Synthesis, evaluation as a class of novel analgesics, and 3D QSAR analysis, Bioorg. Med. Chem., 08/2009, 17 (17), 6305-6310.

5. Yuji Wang, Guifeng Kang, Ming Zhao, Jianhui Wu, Xiaoyi Zhang, Yifan Yang, Jiawang Liu, Shiqi Peng, A new platinum-complex show easy preparation, promising anti-tumor activity, and better efficacy and distribution properties than oxaliplatin, Mol. BioSyst., 12/2011, 7(12), 3245-3252.

6. Ning Li, Guifeng Kang, Lin Gui, Ming Zhao, Wenjing Wang, Jianwei Zhang, Yan-Feng Yue, Shiqi Peng, Novel Cu(II)-RGD-octapeptides: Synthesis, coordination mode, in vitro anti-platelet aggregation/in vivo anti-thrombotic evaluation and correlation of sequence with nano-structure., Nanomed- Nanotechnol., 01/2011, 7(4), 403-409.

7. Yuji Wang, Jianhui Wu, Guifeng Kang, Ming Zhao, Lin Gui,Ning Li, Li Peng, Xiaoyi Zhang, Li Li, Shiqi Peng, Novel nano-materials RGD-tetrapeptide-modified 17β-amino-11α- hydroxyandrost-1,4-diene-3-one: synthesis, self-assembly based nano-images and in vivo anti-osteoporosis evaluation, J.Mater. Chem.,02/2012, 22(11), 4652-4659.

8. Yuji Wang, Jianhui Wu, Guifeng Kang, Ming Zhao, Lin Gui,Ning Li, Li Peng, Xiaoyi Zhang, Li Li, Shiqi Peng, Novel nano-materials RGD-tetrapeptide-modified 17β-amino-11α- hydroxyandrost-1,4-diene-3-one: synthesis, self-assembly based nano-images and in vivo anti-osteoporosis evaluation, J.Mater. Chem.,02/2012, 22(11), 4652-4659.

9. Jingcheng Tang, Ming Zhao, Yuji Wang, Guifeng Kang, Jianhui Wu, Meiqing Zheng, Shiqi Peng, One single HPLC-PDA/(-)ESI-MS/MS analysis to simultaneously determine 30 components of the aqueous extract of Rabdosia rubescens,  J. Chromatogr. B., 09/2011, 879 (26) 2783-2793.

10. Jianhui Wu, Lei Wei, Ming Zhao, Yuji Wang, Guifeng Kang, Shiqi Peng, N-[2(3-Carboxyl-9-benzyl-carboline-1-yl)ethyl-1- yl]-amino acids: correlation of spectral property with in vivo anti-tumor activity, Med. Chem. Res., 04/2012, 21(1), 116-123.

11. Wenjing Wang, Ming Zhao, Yuji Wang, Jiawang Liu, Jianhui Wu, Guifeng Kang and Shiqi Peng, {2-[1-(3-Methoxycarbonylmethyl -1H-indol-2-yl)-1-methyl-ethyl]-1H-indol-3-yl}- acetic acid methyl ester (MIAM): Its anti-cancer efficacy and intercalation mechanism identified via multi-model systems, Mol. BioSyst., 03/2011, 7(3), 766-772.

 

主编或副主编的著作/译著

 

重要奖项

 



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